SCHEMBL4718312

SCHEMBL4718312

Cc1cc(C[CH]C(=O)N2CCC(N3CCN(C(N)=O)CC3)CC2)ccc1Br

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 3/20 0.39
CCR3 P51677 1/20 0.38
ACACB O00763 6/20 0.37
ACACA Q13085 6/20 0.37
GAA P10253 1/20 0.36
ALOX12 P18054 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
L3MBTL3 Q96JM7 5/20 0.36
L3MBTL1 Q9Y468 5/20 0.36
CHRNA3 P32297 1/20 0.36
CHRM2 P08172 1/20 0.35
MBTD1 Q05BQ5 1/20 0.35
MAPT P10636 1/20 0.35
ALDH1A1 P00352 1/20 0.35
POLB P06746 1/20 0.35
HRH3 Q9Y5N1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4717841 1.00 CCR5 (0.39) CCR5CCR3ACACBACACAGAA
SCHEMBL3284870 0.90 CCR5 (0.41) CCR5CCR3ACACBACACAGAA
SCHEMBL3285188 0.90 CCR5 (0.41) CCR5CCR3ACACBACACAGAA
SCHEMBL4717860 0.89 ALDH1A1 (0.39) ALOX12CHRNA3MAPTALDH1A1POLB
SCHEMBL4722465 0.88 CCR3 (0.41) CCR5CCR3ACACBACACAGAA
SCHEMBL3314680 0.88 CCR3 (0.41) CCR5CCR3ACACBACACAGAA
SCHEMBL4717935 0.86 CCR5 (0.36) CCR5CCR3ACACBACACAGAA
SCHEMBL3311181 0.86 CCR5 (0.36) CCR5CCR3ACACBACACAGAA
SCHEMBL3278543 0.85 GAA (0.41) CCR5CCR3ACACBACACAGAA
SCHEMBL3279563 0.83 ACACB (0.38) CCR5ACACBACACAGAAALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1558600-B1 SELECTED CGRP ANTAGONISTS, METHOD FOR PRODUCTION AND USE THEREOF AS MEDICAMENT BOEHRINGER INGELHEIM PHARMA (DE) 2008-05-07 EP claimed