SCHEMBL4718650

SCHEMBL4718650

CS(=O)(=O)c1ccc(-c2cc(C(F)(F)F)nc(Oc3ccc(Br)cc3)n2)cc1

nearest known ligand 0.81

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 11/20 0.81
PTGS2 P35354 12/20 0.65
KDM4E B2RXH2 1/20 0.54
USP2 O75604 1/20 0.54
ALDH1A1 P00352 1/20 0.54
TP53 P04637 1/20 0.54
HPGD P15428 1/20 0.54
KMT2A Q03164 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
NPSR1 Q6W5P4 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4718829 0.89 PTGS1 (1.00) PTGS1PTGS2KDM4EUSP2ALDH1A1
SCHEMBL4718168 0.89 PTGS1 (0.83) PTGS1PTGS2KDM4EUSP2ALDH1A1
SCHEMBL4721120 0.89 PTGS1 (0.83) PTGS1PTGS2KDM4EUSP2ALDH1A1
SCHEMBL4722523 0.85 PTGS1 (0.76) PTGS1PTGS2KDM4EUSP2ALDH1A1
SCHEMBL4722456 0.80 PTGS1 (0.68) PTGS1PTGS2KDM4EUSP2ALDH1A1
SCHEMBL6408442 0.79 PTGS1 (0.67) PTGS1PTGS2KDM4ETP53HPGD
SCHEMBL4504052 0.78 PTGS1 (1.00) PTGS1PTGS2KDM4EUSP2ALDH1A1
SCHEMBL4720953 0.76 PTGS1 (0.48) PTGS1PTGS2
SCHEMBL4721292 0.74 SDHB (0.81) PTGS1PTGS2KDM4EUSP2ALDH1A1
SCHEMBL4720369 0.74 PTGS1 (1.00) PTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1493735-B1 PYRIMIDINE DERIVATIVES USEFUL AS SELECTIVE COX-2 INHIBITORS GLAXO GROUP LTD (GB) 2008-10-29 EP claimed