SCHEMBL4722523

SCHEMBL4722523

CS(=O)(=O)c1ccc(-c2cc(C(F)(F)F)nc(Oc3ccc(F)c(F)c3)n2)cc1

nearest known ligand 0.76

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 12/20 0.76
PTGS2 P35354 11/20 0.64
KDM4E B2RXH2 2/20 0.53
ALDH1A1 P00352 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
NPSR1 Q6W5P4 2/20 0.53
USP2 O75604 1/20 0.53
TP53 P04637 1/20 0.53
HPGD P15428 1/20 0.53
KMT2A Q03164 1/20 0.53
MITF O75030 1/20 0.50
LMNA P02545 1/20 0.50
STAT3 P40763 1/20 0.50
STAT1 P42224 1/20 0.50
RAB9A P51151 1/20 0.50
TLR9 Q9NR96 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4718168 0.88 PTGS1 (0.83) PTGS1PTGS2KDM4EALDH1A1SMN1; SMN2
SCHEMBL4721120 0.86 PTGS1 (0.83) PTGS1PTGS2KDM4EALDH1A1SMN1; SMN2
SCHEMBL4718829 0.86 PTGS1 (1.00) PTGS1PTGS2KDM4EALDH1A1SMN1; SMN2
SCHEMBL4718650 0.85 PTGS1 (0.81) PTGS1PTGS2KDM4EALDH1A1SMN1; SMN2
SCHEMBL4722456 0.81 PTGS1 (0.68) PTGS1PTGS2KDM4EALDH1A1SMN1; SMN2
SCHEMBL6408442 0.78 PTGS1 (0.67) PTGS1PTGS2KDM4ESMN1; SMN2NPSR1
SCHEMBL4504052 0.77 PTGS1 (1.00) PTGS1PTGS2KDM4EALDH1A1SMN1; SMN2
SCHEMBL4718068 0.74 PTGS2 (0.82) PTGS1PTGS2KDM4EALDH1A1SMN1; SMN2
SCHEMBL4721292 0.73 SDHB (0.81) PTGS1PTGS2KDM4EALDH1A1SMN1; SMN2
SCHEMBL4720369 0.73 PTGS1 (1.00) PTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1493735-B1 PYRIMIDINE DERIVATIVES USEFUL AS SELECTIVE COX-2 INHIBITORS GLAXO GROUP LTD (GB) 2008-10-29 EP claimed