SCHEMBL4724504

SCHEMBL4724504

COc1cc(-c2nn(-c3cc(N4CCC(O)C4)ccc3C(F)(F)F)c(=O)c3[nH]ccc23)ccc1F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 2/20 0.38
ICAM1 P05362 2/20 0.38
ITGAL P20701 2/20 0.38
PDE7A Q13946 2/20 0.36
MCHR1 Q99705 2/20 0.36
RORC P51449 1/20 0.36
PDE3B Q13370 3/20 0.35
PDE3A Q14432 3/20 0.35
SMPD3 Q9NY59 3/20 0.35
ROCK2 O75116 1/20 0.34
P2RX7 Q99572 1/20 0.34
NOTUM Q6P988 1/20 0.34
MAPT P10636 1/20 0.33
CACNA2D1 P54289 1/20 0.33
GAK O14976 1/20 0.33
INSR P06213 1/20 0.33
IGF1R P08069 1/20 0.33
INSRR P14616 1/20 0.33
MAPK1 P28482 1/20 0.33
LTK P29376 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4724501 1.00 ITGB2 (0.38) ITGB2ICAM1ITGALPDE7AMCHR1
SCHEMBL4765817 0.90 P2RX7 (0.38) RORCPDE3BPDE3AP2RX7NOTUM
SCHEMBL4765812 0.90 P2RX7 (0.38) RORCPDE3BPDE3AP2RX7NOTUM
SCHEMBL4718873 0.90 P2RX7 (0.35) ITGB2ICAM1ITGALPDE7ARORC
SCHEMBL4718877 0.90 P2RX7 (0.35) ITGB2ICAM1ITGALPDE7ARORC
SCHEMBL14102050 0.89 PDE10A (0.37) ROCK2NOTUMMAPTMAPK1
SCHEMBL4722458 0.85 ABL1 (0.39) ITGB2ICAM1ITGALPDE7ARORC
SCHEMBL4722453 0.85 ABL1 (0.39) ITGB2ICAM1ITGALPDE7ARORC
SCHEMBL4723372 0.84 PDE4A (0.43) ITGB2ICAM1ITGALPDE7AMCHR1
SCHEMBL4723378 0.84 PDE4A (0.43) ITGB2ICAM1ITGALPDE7AMCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed