SCHEMBL4718934

SCHEMBL4718934

COc1cc(OC)cc(-c2nn(-c3cc(N4CCC(C(=O)O)C4)ccc3C(F)(F)F)c(=O)c3c2CCC3)c1

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 16/20 0.47
S1PR1 P21453 1/20 0.40
NEK2 P51955 1/20 0.37
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
UGCG Q16739 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4722716 0.93 NOTUM (0.38) NOTUMS1PR1PDE4APDE4BPDE4C
SCHEMBL4723394 0.93 HSD11B1 (0.39) NOTUMS1PR1PDE4APDE4BPDE4C
SCHEMBL4719376 0.92 NOTUM (0.49) NOTUMS1PR1PDE4APDE4BPDE4C
SCHEMBL4722787 0.92 NOTUM (0.48) NOTUMS1PR1PDE4APDE4BPDE4C
SCHEMBL4722706 0.92 NOTUM (0.48) NOTUMS1PR1PDE4APDE4BPDE4C
SCHEMBL4721983 0.90 NOTUM (0.40) NOTUMS1PR1UGCG
SCHEMBL4721118 0.90 NOTUM (0.43) NOTUM
SCHEMBL4719501 0.90 P2RX7 (0.38) PDE4APDE4BPDE4CPDE4DUGCG
SCHEMBL4719498 0.90 P2RX7 (0.38) PDE4APDE4BPDE4CPDE4DUGCG
SCHEMBL4724695 0.90 P2RX7 (0.38) PDE4APDE4BPDE4CPDE4DUGCG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed