SCHEMBL4718995

SCHEMBL4718995

Cc1ccc(NC(=O)NCc2cc(CN3CCN(C(C)(C)C)CC3)ccc2F)cn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 6/20 0.41
KCNQ3 O43525 1/20 0.40
KCNQ2 O43526 1/20 0.40
GALR3 O60755 1/20 0.39
RAB9A P51151 1/20 0.39
CHRM1 P11229 1/20 0.39
HTR2A P28223 1/20 0.39
MCHR1 Q99705 1/20 0.39
TRPV1 Q8NER1 2/20 0.38
FAAH O00519 3/20 0.38
NPY2R P49146 1/20 0.38
WNT1 P04628 1/20 0.38
CLK2 P49760 1/20 0.38
CLK3 P49761 1/20 0.38
DYRK1A Q13627 1/20 0.38
ACKR3 P25106 1/20 0.37
TP53 P04637 1/20 0.37
MAPT P10636 1/20 0.37
CHRNA7 P36544 1/20 0.37
ALOX5 P09917 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3732394 0.90 FAAH (0.41) NAMPTKCNQ3KCNQ2CHRM1HTR2A
SCHEMBL4709225 0.89 NAMPT (0.43) NAMPTRAB9ACHRM1HTR2AMCHR1
SCHEMBL3728465 0.88 MEN1 (0.43) NAMPTKCNQ3KCNQ2CHRM1HTR2A
SCHEMBL3735920 0.87 TBK1 (0.45) NAMPTFAAHMAPTEPHX2
SCHEMBL3733024 0.87 NAMPT (0.47) NAMPTKCNQ3KCNQ2TRPV1
SCHEMBL3738335 0.87 PIK3CA (0.47) NAMPTTRPV1
SCHEMBL3733287 0.87 FAAH (0.41) NAMPTKCNQ3KCNQ2CHRM1HTR2A
SCHEMBL3742347 0.87 FAAH (0.41) NAMPTKCNQ3KCNQ2GALR3RAB9A
SCHEMBL3744319 0.86 ALDH1A1 (0.47) NAMPTFAAH
SCHEMBL3742331 0.84 NAMPT (0.45) NAMPTKCNQ3KCNQ2TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1959947-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS AND METHODS Cytokinetics, Inc. (US) 2008-08-27 EP disclosed
WO-2007075377-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS AND METHODS CYTOKINETICS, INC. (US) 2007-07-05 WO disclosed