SCHEMBL4720175

SCHEMBL4720175

CC(C)(C)OC(=O)ON1CCc2c(c3cc(Br)ccc3n2CC(=O)O)C1

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KRAS P01116 4/20 0.51
BAZ2B Q9UIF8 2/20 0.48
AKR1B10 O60218 2/20 0.47
AKR1B1 P15121 2/20 0.47
PTGDR2 Q9Y5Y4 7/20 0.46
HDAC1 Q13547 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
AKR1A1 P14550 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4719430 0.89 PTGDR2 (0.59) BAZ2BAKR1B10AKR1B1PTGDR2HDAC1
SCHEMBL4719539 0.88 PTGDR2 (0.58) BAZ2BPTGDR2
SCHEMBL4721545 0.88 BAZ2B (0.64) BAZ2BAKR1B10AKR1B1PTGDR2HDAC1
SCHEMBL3085456 0.85 KRAS (0.67) KRASBAZ2BAKR1B10AKR1B1PTGDR2
SCHEMBL4721439 0.83 PTGDR2 (0.59) BAZ2BAKR1B10AKR1B1PTGDR2HDAC1
SCHEMBL4722882 0.82 BAZ2B (0.53) BAZ2BAKR1B10AKR1B1PTGDR2AKR1A1
SCHEMBL4718940 0.77 PTGDR2 (0.60) BAZ2BPTGDR2HDAC1HDAC6
SCHEMBL3083804 0.74 PTGDR2 (0.68) KRASBAZ2BAKR1B10AKR1B1PTGDR2
SCHEMBL5026847 0.73 TSPO (0.39) KRAS
SCHEMBL3096312 0.73 PTGDR2 (0.77) PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1725553-B1 TETRAHYDROPYRIDOINDOLE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2008-05-07 EP claimed