SCHEMBL4720286

SCHEMBL4720286

Cc1cc(C)cc(-c2nn(-c3cc(-c4cccnn4)ccc3C(F)(F)F)c(=O)c3c2CC(C)N3)c1

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.32
CREBBP Q92793 1/20 0.32
P2RX7 Q99572 1/20 0.32
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4723868 0.93 BRD4 (0.31) BRD4CREBBP
SCHEMBL4721734 0.92 P2RX7 (0.31) P2RX7SLC6A2SLC6A4SLC6A3
SCHEMBL4721383 0.90 BRD4 (0.32) BRD4CREBBPP2RX7
SCHEMBL4719906 0.90 BRD4 (0.34) BRD4CREBBP
SCHEMBL4721949 0.86 NTRK1 (0.33) SLC6A2SLC6A4SLC6A3
SCHEMBL4723419 0.84 MEN1 (0.31)
SCHEMBL4724001 0.83 PDE4A (0.36) P2RX7
SCHEMBL4719842 0.83 PDE4A (0.38) P2RX7
SCHEMBL4720712 0.83
SCHEMBL4721524 0.83 BRD4 (0.33) BRD4CREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed