SCHEMBL4719906

SCHEMBL4719906

COc1cc(OC)cc(-c2nn(-c3cc(-c4cccnn4)ccc3C(F)(F)F)c(=O)c3c2CC(C)N3)c1

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.34
CREBBP Q92793 1/20 0.34
GRM7 Q14831 1/20 0.32
CCNA2 P20248 1/20 0.31
CDK2 P24941 1/20 0.31
CCNA1 P78396 1/20 0.31
CYP11B1 P15538 1/20 0.30
CYP11B2 P19099 1/20 0.30
SYK P43405 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4723868 0.96 BRD4 (0.31) BRD4CREBBPGRM7
SCHEMBL4720286 0.90 BRD4 (0.32) BRD4CREBBP
SCHEMBL4724951 0.87 NTRK1 (0.32) GRM7
SCHEMBL4765008 0.82 NTRK1 (0.31)
SCHEMBL4721383 0.82 BRD4 (0.32) BRD4CREBBP
SCHEMBL4721734 0.82 P2RX7 (0.31)
SCHEMBL4723635 0.80 PDE4A (0.38) GRM7
SCHEMBL4724223 0.77 PDE3B (0.36)
SCHEMBL4724224 0.77 PDE3B (0.36)
SCHEMBL4721949 0.76 NTRK1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed