SCHEMBL4720739

SCHEMBL4720739

CC[C@@H](NC(C)=O)c1nc(-c2ccc(C[C@@H](CCO)NC(=O)c3ccc(OC(C)C)c(Cl)c3)cc2)c(C)[nH]1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CENPE Q02224 3/20 0.45
KIFC1 Q9BW19 1/20 0.38
TOP2A P11388 1/20 0.37
TAS1R3 Q7RTX0 4/20 0.36
TAS1R1 Q7RTX1 4/20 0.36
S1PR1 P21453 2/20 0.35
S1PR3 Q99500 1/20 0.35
S1PR5 Q9H228 1/20 0.35
FOXO1 Q12778 1/20 0.34
F11 P03951 1/20 0.34
PRSS1 P07477 1/20 0.34
PRSS2 P07478 1/20 0.34
PRSS3 P35030 1/20 0.34
MME P08473 2/20 0.33
MAP4K4 O95819 1/20 0.33
MINK1 Q8N4C8 1/20 0.33
ROCK2 O75116 1/20 0.33
PRKACA P17612 1/20 0.33
RPS6KB1 P23443 1/20 0.33
IRAK1 P51617 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4717914 0.86 CENPE (0.42) CENPEKIFC1TOP2ATAS1R3TAS1R1
SCHEMBL3229213 0.81 CENPE (0.51) CENPEKIFC1TAS1R3TAS1R1S1PR1
SCHEMBL3461569 0.81 CENPE (0.51) CENPEKIFC1TAS1R3TAS1R1S1PR1
SCHEMBL13161447 0.81 CENPE (0.51) CENPEKIFC1TAS1R3TAS1R1S1PR1
SCHEMBL4722632 0.80 CENPE (0.42) CENPEKIFC1TOP2ATAS1R3TAS1R1
SCHEMBL4720522 0.80 CENPE (0.43) CENPEKIFC1TOP2ATAS1R3TAS1R1
SCHEMBL13644414 0.79 CENPE (0.47) CENPEKIFC1TOP2ATAS1R3TAS1R1
SCHEMBL4718875 0.78 CENPE (0.45) CENPEKIFC1TOP2ATAS1R3TAS1R1
SCHEMBL3219624 0.77 CENPE (0.52) CENPEKIFC1TAS1R3TAS1R1S1PR1
SCHEMBL2104729 0.77 SIRT2 (0.46) CENPEKIFC1TAS1R3TAS1R1PKN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1951719-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS Cytokinetics, Inc. (US) 2008-08-06 EP disclosed
WO-2007056469-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INC. (US) 2007-05-18 WO disclosed