SCHEMBL4720845

SCHEMBL4720845

COc1cc(-c2nn(-c3cc(N4CC(CO)C4)ccc3C(F)(F)F)c(=O)c3c2CCN3CCO)ccc1F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
KCNK3 O14649 2/20 0.33
ALK Q9UM73 2/20 0.31
HTR2C P28335 1/20 0.31
CACNA2D1 P54289 1/20 0.31
ROCK2 O75116 2/20 0.31
ITGB2 P05107 1/20 0.31
ICAM1 P05362 1/20 0.31
ITGAL P20701 1/20 0.31
TGFBR1 P36897 1/20 0.31
ACVR1 Q04771 1/20 0.31
KCNH2 Q12809 1/20 0.31
GRM2 Q14416 2/20 0.31
KDM1A O60341 2/20 0.31
CCR1 P32246 1/20 0.30
UGCG Q16739 1/20 0.30
CXCR3 P49682 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4718895 0.91 CYP3A4 (0.32)
SCHEMBL4724276 0.90 ITGB2 (0.35) PDE4APDE4BPDE4CPDE4DKCNK3
SCHEMBL4724274 0.90 ITGB2 (0.35) PDE4APDE4BPDE4CPDE4DKCNK3
SCHEMBL4723157 0.90 F10 (0.32) CCR1CXCR3LGALS3
SCHEMBL4722298 0.89 PDE4A (0.35) PDE4APDE4BPDE4CPDE4DKCNK3
SCHEMBL4719683 0.88 SMN1; SMN2 (0.34) PDE4APDE4BPDE4CPDE4DKCNK3
SCHEMBL4766343 0.87 F10 (0.31) CXCR3
SCHEMBL4722273 0.87 SMPD3 (0.45) ITGB2ICAM1ITGAL
SCHEMBL4722270 0.87 SMPD3 (0.45) ITGB2ICAM1ITGAL
SCHEMBL4724909 0.86 PDE4A (0.32) PDE4APDE4BPDE4CPDE4DUGCG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed