SCHEMBL4718895

SCHEMBL4718895

Cc1cc(-c2nn(-c3cc(N4CC(CO)C4)ccc3C(F)(F)F)c(=O)c3c2CCN3CCO)ccc1F

nearest known ligand 0.32

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
C5AR1 P21730 1/20 0.30
SYK P43405 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4720845 0.91 PDE4A (0.36)
SCHEMBL4718914 0.90 P2RX7 (0.36) CYP3A4CYP2C9NPSR1
SCHEMBL4724182 0.90 P2RX7 (0.36) CYP3A4CYP2C9NPSR1
SCHEMBL4718912 0.90 P2RX7 (0.36) CYP3A4CYP2C9NPSR1
SCHEMBL4722697 0.89 CYP3A4 (0.35) CYP3A4CYP2C9NPSR1
SCHEMBL4720993 0.88
SCHEMBL4720752 0.87 LGALS3 (0.34)
SCHEMBL4723157 0.86 F10 (0.32)
SCHEMBL4719683 0.85 SMN1; SMN2 (0.34) CYP2C9
SCHEMBL4766343 0.83 F10 (0.31) CYP3A4CYP2C9NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed