SCHEMBL4721877

SCHEMBL4721877

COc1cccc(-c2cc(NC(=O)O)c(=O)n(-c3cc(N4CCOCC4)ccn3)n2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
NPC1 O15118 3/20 0.44
RAB9A P51151 3/20 0.44
MTOR P42345 1/20 0.44
SMG1 Q96Q15 1/20 0.44
CCNT1 O60563 1/20 0.42
CDK9 P50750 1/20 0.42
STK4 Q13043 1/20 0.41
STK3 Q13188 1/20 0.41
LRRK2 Q5S007 1/20 0.41
DGAT1 O75907 1/20 0.41
SOAT1 P35610 1/20 0.41
CYP1A2 P05177 2/20 0.41
CYP1A1 P04798 1/20 0.41
CYP1B1 Q16678 1/20 0.41
ALDH1A1 P00352 2/20 0.41
LMNA P02545 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
USP2 O75604 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14101818 0.90 MEN1 (0.46) MEN1KMT2ANPC1RAB9AMTOR
SCHEMBL4722479 0.87 MTOR (0.45) MEN1KMT2ANPC1RAB9AMTOR
SCHEMBL4721933 0.85 MTOR (0.45) MEN1KMT2ANPC1RAB9AMTOR
SCHEMBL4720924 0.85 DGAT1 (0.48) MEN1KMT2AMTORSMG1CCNT1
SCHEMBL4722075 0.73 MEN1 (0.47) MEN1KMT2ACYP1A2CYP1A1CYP1B1
SCHEMBL14101741 0.73 MEN1 (0.46) MEN1KMT2ASTK4STK3LRRK2
SCHEMBL4722685 0.73 MEN1 (0.46) MEN1KMT2ANPC1RAB9ACCNT1
SCHEMBL4719536 0.72 MAPT (0.51) MEN1KMT2ACYP1A2CYP1A1CYP1B1
SCHEMBL4724315 0.72 MEN1 (0.45) MEN1KMT2ANPC1RAB9ASTK4
SCHEMBL4719650 0.72 PRKDC (0.48) MEN1KMT2ANPC1RAB9ASTK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed