SCHEMBL4721933

SCHEMBL4721933

COc1cccc(-c2cc(N)c(=O)n(-c3cc(N4CCOCC4)ccn3)n2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTOR P42345 1/20 0.45
SMG1 Q96Q15 1/20 0.45
STK4 Q13043 1/20 0.44
STK3 Q13188 1/20 0.44
LRRK2 Q5S007 1/20 0.44
PRKDC P78527 1/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
CYP1A2 P05177 3/20 0.43
CYP3A4 P08684 2/20 0.43
TSHR P16473 2/20 0.43
MAPK1 P28482 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP2C9 P11712 1/20 0.43
HSD17B10 Q99714 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
PIK3CA P42336 1/20 0.42
GSK3B P49841 1/20 0.42
GAK O14976 1/20 0.42
CYP1A1 P04798 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4722479 0.86 MTOR (0.45) MTORSMG1STK4STK3LRRK2
SCHEMBL4721877 0.85 MEN1 (0.47) MTORSMG1STK4STK3LRRK2
SCHEMBL4720924 0.83 DGAT1 (0.48) MTORSMG1MEN1KMT2AL3MBTL1
SCHEMBL14101818 0.82 MEN1 (0.46) MTORSMG1STK4STK3LRRK2
SCHEMBL4722809 0.76 GAA (0.54) STK4STK3LRRK2PRKDCMEN1
SCHEMBL4719650 0.75 PRKDC (0.48) STK4STK3LRRK2PRKDCMEN1
SCHEMBL4723995 0.75 GAA (0.50) STK4STK3LRRK2PRKDCMEN1
SCHEMBL4723982 0.74 GAA (0.51) STK4STK3LRRK2PRKDCMEN1
SCHEMBL4764880 0.72 PRKDC (0.43) STK4STK3LRRK2PRKDCMEN1
SCHEMBL14101741 0.71 MEN1 (0.46) STK4STK3LRRK2PRKDCMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed