SCHEMBL4722067

SCHEMBL4722067

COc1cc(OC)cc(-c2cn(-c3cc(N4CC[C@H](O)C4)ccc3C(F)(F)F)c(=O)c3c2CCC3)c1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.39
PDE7A Q13946 1/20 0.35
MCHR1 Q99705 2/20 0.34
HSD11B1 P28845 3/20 0.34
F10 P00742 2/20 0.34
F2 P00734 1/20 0.34
PDE3B Q13370 2/20 0.34
PDE3A Q14432 2/20 0.34
ABL1 P00519 1/20 0.34
NOTUM Q6P988 1/20 0.33
ITGB2 P05107 1/20 0.33
ICAM1 P05362 1/20 0.33
ITGAL P20701 1/20 0.33
S1PR1 P21453 1/20 0.33
SOS1 Q07889 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4722070 1.00 P2RX7 (0.39) P2RX7PDE7AMCHR1HSD11B1F10
SCHEMBL14102092 0.91 PDK2 (0.34) NOTUMS1PR1
SCHEMBL14101726 0.88 F2 (0.37) P2RX7F10F2NOTUMS1PR1
SCHEMBL4720703 0.88 ITGB2 (0.39) ITGB2ICAM1ITGAL
SCHEMBL4720700 0.88 ITGB2 (0.39) ITGB2ICAM1ITGAL
SCHEMBL4718933 0.87 P2RX7 (0.38) P2RX7PDE7AMCHR1HSD11B1F10
SCHEMBL4718937 0.87 P2RX7 (0.38) P2RX7PDE7AMCHR1HSD11B1F10
SCHEMBL4724969 0.86 NOTUM (0.36) NOTUMS1PR1
SCHEMBL4722470 0.86 NOTUM (0.36) NOTUMS1PR1
SCHEMBL4722462 0.86 NOTUM (0.36) NOTUMS1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed