SCHEMBL4722202

SCHEMBL4722202

CC(=O)N1CCCc2c(-c3cc(C)cc(-c4cnco4)c3)nn(-c3c(Cl)cccc3Cl)c(=O)c21

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CREBBP Q92793 3/20 0.36
NOTUM Q6P988 2/20 0.35
CYP11B2 P19099 6/20 0.34
BRD4 O60885 2/20 0.33
IMPDH2 P12268 2/20 0.33
P2RY1 P47900 1/20 0.32
RHOA P61586 1/20 0.32
NPSR1 Q6W5P4 1/20 0.31
LIMK2 P53671 1/20 0.31
LMNA P02545 1/20 0.31
TP53 P04637 1/20 0.31
BACE1 P56817 2/20 0.30
BACE2 Q9Y5Z0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4719705 0.88 BACE1 (0.33) CREBBPIMPDH2P2RY1RHOALMNA
SCHEMBL4722893 0.87 CREBBP (0.32) CREBBPIMPDH2P2RY1RHOALIMK2
SCHEMBL4719544 0.86 CNR1 (0.33) CREBBPBACE1BACE2
SCHEMBL4765691 0.86 CREBBP (0.32) CREBBPIMPDH2BACE1BACE2
SCHEMBL4721258 0.85 BACE1 (0.30) BACE1BACE2
SCHEMBL4723886 0.85 P2RY1 (0.33) CREBBPIMPDH2P2RY1RHOALIMK2
SCHEMBL14101802 0.84
SCHEMBL4723382 0.84 ACHE (0.34) CREBBPP2RY1LMNATP53
SCHEMBL4723733 0.83 BACE1 (0.31) CREBBPBACE1BACE2
SCHEMBL4720247 0.81 BACE1 (0.32) IMPDH2P2RY1LMNABACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed