SCHEMBL4765691

SCHEMBL4765691

Cc1cc(-c2cnco2)cc(-c2nn(-c3c(Cl)cccc3Cl)c(=O)c3c2CCCN3CCO)c1

nearest known ligand 0.32

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CREBBP Q92793 1/20 0.32
USP7 Q93009 2/20 0.31
BACE1 P56817 1/20 0.31
BACE2 Q9Y5Z0 1/20 0.31
IMPDH2 P12268 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4723733 0.92 BACE1 (0.31) CREBBPBACE1BACE2
SCHEMBL4719544 0.91 CNR1 (0.33) CREBBPBACE1BACE2
SCHEMBL4722893 0.90 CREBBP (0.32) CREBBPIMPDH2
SCHEMBL14101802 0.89
SCHEMBL4719705 0.89 BACE1 (0.33) CREBBPUSP7BACE1BACE2IMPDH2
SCHEMBL4723886 0.88 P2RY1 (0.33) CREBBPIMPDH2
SCHEMBL4723382 0.87 ACHE (0.34) CREBBP
SCHEMBL4722202 0.86 CREBBP (0.36) CREBBPBACE1BACE2IMPDH2
SCHEMBL4721258 0.84 BACE1 (0.30) BACE1BACE2
SCHEMBL4720247 0.80 BACE1 (0.32) BACE1BACE2IMPDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed