SCHEMBL4722249

SCHEMBL4722249

Cc1cc(C)cc(-c2nn(-c3cc(N4CCC(O)C4)ccc3C(F)(F)F)c(=O)c3c2CCN3C(N)=O)c1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.38
PDE3B Q13370 2/20 0.33
PDE3A Q14432 2/20 0.33
NOTUM Q6P988 5/20 0.33
RORC P51449 1/20 0.33
HSD11B1 P28845 3/20 0.32
SOS1 Q07889 2/20 0.32
MYC P01106 2/20 0.32
WDR5 P61964 2/20 0.32
PHGDH O43175 1/20 0.32
LCK P06239 1/20 0.32
JAK3 P52333 1/20 0.32
F10 P00742 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4722245 1.00 P2RX7 (0.38) P2RX7PDE3BPDE3ANOTUMRORC
SCHEMBL4724414 0.90 P2RX7 (0.35) P2RX7PDE3BPDE3ANOTUMRORC
SCHEMBL4724420 0.90 P2RX7 (0.35) P2RX7PDE3BPDE3ANOTUMRORC
SCHEMBL4720193 0.89 SMPD3 (0.38)
SCHEMBL4720195 0.89 SMPD3 (0.38)
SCHEMBL4724669 0.89 MAPT (0.35) P2RX7NOTUMWDR5F10
SCHEMBL4720477 0.89 P2RX7 (0.37) P2RX7PDE3BPDE3ANOTUMRORC
SCHEMBL4720480 0.89 P2RX7 (0.37) P2RX7PDE3BPDE3ANOTUMRORC
SCHEMBL4720304 0.88 SMPD3 (0.35) P2RX7NOTUMRORCMYCWDR5
SCHEMBL4720300 0.88 SMPD3 (0.35) P2RX7NOTUMRORCMYCWDR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed