SCHEMBL4722512

SCHEMBL4722512

Cc1cc(-c2cnco2)cc(-c2nn(-c3cc(Br)ccc3F)c(=O)c3ccccc23)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 8/20 0.38
MAPT P10636 3/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.35
GAA P10253 4/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
LMNA P02545 4/20 0.34
ALDH1A1 P00352 3/20 0.32
KDM4E B2RXH2 2/20 0.32
PDE4A P27815 1/20 0.32
PDE4B Q07343 1/20 0.32
PDE4C Q08493 1/20 0.32
PDE4D Q08499 1/20 0.32
PKM P14618 1/20 0.32
CYP1A2 P05177 2/20 0.32
CYP2C9 P11712 2/20 0.32
CYP2C19 P33261 2/20 0.32
CYP3A4 P08684 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4719884 0.87 L3MBTL1 (0.36) NPSR1MAPTMEN1KMT2AL3MBTL1
SCHEMBL4721927 0.87 ALOX5 (0.37) NPSR1MAPTMEN1KMT2AL3MBTL1
SCHEMBL4719229 0.85 IMPDH2 (0.40) NPSR1MAPTNPC1RAB9ALMNA
SCHEMBL4723560 0.83 MAPT (0.39) NPSR1MAPTMEN1KMT2AGAA
SCHEMBL4722439 0.78 MEN1 (0.43) NPSR1MAPTMEN1KMT2AGAA
SCHEMBL4721167 0.78 NPSR1 (0.43) NPSR1MAPTMEN1KMT2AL3MBTL1
SCHEMBL4719649 0.78 MEN1 (0.40) NPSR1MAPTMEN1KMT2AGAA
SCHEMBL4719701 0.78 GAA (0.41) NPSR1MAPTMEN1KMT2AL3MBTL1
SCHEMBL4722197 0.78 MEN1 (0.32) MEN1KMT2AGAA
SCHEMBL4719136 0.78 MAPT (0.37) NPSR1MAPTMEN1KMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed