SCHEMBL4722609

SCHEMBL4722609

COc1cncc(-c2nn(-c3cc(N4CC[C@H](O)C4)ccc3C(F)(F)F)c(=O)c3c2CCN3C(N)=O)c1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 1/20 0.39
CYP11B2 P19099 5/20 0.34
P2RX7 Q99572 1/20 0.34
CYP11B1 P15538 3/20 0.34
CHRNB2 P17787 2/20 0.33
CHRNB4 P30926 2/20 0.33
CHRNA3 P32297 2/20 0.33
CHRNA4 P43681 2/20 0.33
F10 P00742 6/20 0.33
F2 P00734 2/20 0.33
HTR2A P28223 3/20 0.32
HTR2C P28335 3/20 0.32
HTR2B P41595 3/20 0.32
CYP1A2 P05177 3/20 0.32
RPS6KB1 P23443 1/20 0.32
HSP90AA1 P07900 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4722615 1.00 ABL1 (0.39) ABL1CYP11B2P2RX7CYP11B1CHRNB2
SCHEMBL4724414 0.93 P2RX7 (0.35) ABL1P2RX7F10F2
SCHEMBL4724420 0.93 P2RX7 (0.35) ABL1P2RX7F10F2
SCHEMBL4721854 0.91 P2RX7 (0.37) P2RX7F10F2
SCHEMBL4721851 0.91 P2RX7 (0.37) P2RX7F10F2
SCHEMBL4719240 0.88 ABL1 (0.38) ABL1CYP11B2P2RX7CYP11B1CHRNB2
SCHEMBL4719238 0.88 ABL1 (0.38) ABL1CYP11B2P2RX7CYP11B1CHRNB2
SCHEMBL4722192 0.87 CYP11B2 (0.32) CYP11B2CYP11B1
SCHEMBL4722194 0.87 CYP11B2 (0.32) CYP11B2CYP11B1
SCHEMBL4722193 0.87 CYP11B2 (0.32) CYP11B2CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed