SCHEMBL4722958

SCHEMBL4722958

COc1cc(C)cc(-c2nn(-c3cc(N4CC[C@@H](O)C4)ccc3C(F)(F)F)c(=O)c3c2CCC3)c1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.38
F10 P00742 6/20 0.35
F2 P00734 1/20 0.35
UGCG Q16739 1/20 0.35
PDE7A Q13946 1/20 0.35
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35
SOS1 Q07889 2/20 0.34
ROS1 P08922 1/20 0.34
PDE3B Q13370 2/20 0.33
PDE3A Q14432 2/20 0.33
ITGB2 P05107 1/20 0.33
ICAM1 P05362 1/20 0.33
ITGAL P20701 1/20 0.33
FFAR1 O14842 1/20 0.32
HSD11B1 P28845 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4719627 1.00 P2RX7 (0.38) P2RX7F10F2UGCGPDE7A
SCHEMBL4719624 1.00 P2RX7 (0.38) P2RX7F10F2UGCGPDE7A
SCHEMBL4724695 0.95 P2RX7 (0.38) P2RX7F10F2UGCGPDE7A
SCHEMBL4719498 0.95 P2RX7 (0.38) P2RX7F10F2UGCGPDE7A
SCHEMBL4719501 0.95 P2RX7 (0.38) P2RX7F10F2UGCGPDE7A
SCHEMBL4766334 0.93 P2RX7 (0.41) P2RX7PDE7ASOS1PDE3BPDE3A
SCHEMBL4766349 0.93 P2RX7 (0.41) P2RX7PDE7ASOS1PDE3BPDE3A
SCHEMBL4718755 0.92 ROCK2 (0.37) P2RX7F10F2UGCGPDE7A
SCHEMBL4718757 0.92 ROCK2 (0.37) P2RX7F10F2UGCGPDE7A
SCHEMBL4766656 0.92 P2RX7 (0.36) P2RX7F10F2UGCGPDE7A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed