SCHEMBL4718757

SCHEMBL4718757

COc1cc(F)cc(-c2nn(-c3cc(N4CCC(O)C4)ccc3C(F)(F)F)c(=O)c3c2CCC3)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 2/20 0.37
P2RX7 Q99572 1/20 0.37
LRRK2 Q5S007 1/20 0.36
HSD11B1 P28845 3/20 0.35
F10 P00742 3/20 0.35
F2 P00734 1/20 0.35
UGCG Q16739 1/20 0.35
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35
HRH3 Q9Y5N1 1/20 0.34
PDE3B Q13370 2/20 0.33
PDE3A Q14432 2/20 0.33
PDE7A Q13946 1/20 0.33
OPRM1 P35372 1/20 0.33
CACNA2D1 P54289 1/20 0.33
ITGB2 P05107 1/20 0.33
ICAM1 P05362 1/20 0.33
ITGAL P20701 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4718755 1.00 ROCK2 (0.37) ROCK2P2RX7LRRK2HSD11B1F10
SCHEMBL4724695 0.95 P2RX7 (0.38) P2RX7HSD11B1F10F2UGCG
SCHEMBL4719501 0.95 P2RX7 (0.38) P2RX7HSD11B1F10F2UGCG
SCHEMBL4719498 0.95 P2RX7 (0.38) P2RX7HSD11B1F10F2UGCG
SCHEMBL4719627 0.92 P2RX7 (0.38) P2RX7HSD11B1F10F2UGCG
SCHEMBL4719624 0.92 P2RX7 (0.38) P2RX7HSD11B1F10F2UGCG
SCHEMBL4722958 0.92 P2RX7 (0.38) P2RX7HSD11B1F10F2UGCG
SCHEMBL4766656 0.92 P2RX7 (0.36) P2RX7HSD11B1F10F2UGCG
SCHEMBL4766649 0.92 P2RX7 (0.36) P2RX7HSD11B1F10F2UGCG
SCHEMBL4720188 0.91 PTGS2 (0.40) P2RX7F10F2UGCGPDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed