SCHEMBL4722983

SCHEMBL4722983

COc1cc(OC)cc(-c2nn(-c3cc(N4CC[C@H](O)C4)ccc3C(F)(F)F)c(=O)c3c2CCN3CC(=O)N2CCN(C)CC2)c1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.36
CCR1 P32246 7/20 0.35
F10 P00742 6/20 0.34
F2 P00734 1/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
CXCR3 P49682 2/20 0.33
SLC6A9 P48067 1/20 0.33
CYP2C19 P33261 1/20 0.33
KCNH2 Q12809 1/20 0.33
OPRM1 P35372 1/20 0.32
CACNA2D1 P54289 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4722990 1.00 P2RX7 (0.36) P2RX7CCR1F10F2NPC1
SCHEMBL4719634 0.96 F10 (0.37) P2RX7CCR1F10F2CXCR3
SCHEMBL4719639 0.96 F10 (0.37) P2RX7CCR1F10F2CXCR3
SCHEMBL4719706 0.95 P2RX7 (0.35) P2RX7CCR1F10F2CXCR3
SCHEMBL4719710 0.95 P2RX7 (0.35) P2RX7CCR1F10F2CXCR3
SCHEMBL4721375 0.95 F10 (0.34) P2RX7CCR1F10F2CXCR3
SCHEMBL4721377 0.95 F10 (0.34) P2RX7CCR1F10F2CXCR3
SCHEMBL4724775 0.94 NOTUM (0.35) P2RX7CCR1F10F2NPC1
SCHEMBL4724779 0.94 NOTUM (0.35) P2RX7CCR1F10F2NPC1
SCHEMBL4720618 0.91 F10 (0.36) P2RX7F10F2CXCR3SLC6A9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed