SCHEMBL4723153

SCHEMBL4723153

Cc1cc(C)cc(-c2nn(-c3cc(Br)ccc3C(F)(F)F)c(=O)c3c2CCN3)c1

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 1/20 0.33
PARP10 Q53GL7 2/20 0.31
PARP11 Q9NR21 2/20 0.31
PARP15 Q460N3 1/20 0.31
PARP14 Q460N5 1/20 0.31
TIPARP Q7Z3E1 1/20 0.31
PARP16 Q8N5Y8 1/20 0.31
LMNA P02545 1/20 0.31
HCAR1 Q9BXC0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4719266 0.88 LRRK2 (0.33) NTRK1
SCHEMBL4721949 0.83 NTRK1 (0.33) NTRK1
SCHEMBL4721524 0.83 BRD4 (0.33)
SCHEMBL4723711 0.80 P2RX7 (0.38)
SCHEMBL4723707 0.80 P2RX7 (0.38)
SCHEMBL4723419 0.78 MEN1 (0.31)
SCHEMBL4722852 0.77 GRIN1 (0.34) NTRK1
SCHEMBL4720876 0.77 CYP11B1 (0.33) NTRK1
SCHEMBL4765008 0.77 NTRK1 (0.31) NTRK1
SCHEMBL4764976 0.77 CNR1 (0.34) NTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed