SCHEMBL4720876

SCHEMBL4720876

COc1cc(OC)cc(-c2nn(-c3cc(F)ccc3C(F)(F)F)c(=O)c3c2CCN3)c1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 2/20 0.33
CYP11B2 P19099 2/20 0.33
LRRK2 Q5S007 1/20 0.33
RIPK3 Q9Y572 2/20 0.33
GRM7 Q14831 1/20 0.33
WDR5 P61964 1/20 0.32
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 2/20 0.32
HPGD P15428 2/20 0.32
ALPL P05186 1/20 0.32
ALPI P09923 1/20 0.32
NTRK1 P04629 1/20 0.32
HTR2A P28223 2/20 0.31
HTR2C P28335 2/20 0.31
HTR2B P41595 2/20 0.31
GRIN1 Q05586 1/20 0.30
GRIN2B Q13224 1/20 0.30
MAPT P10636 1/20 0.30
MTNR1A P48039 1/20 0.30
MTNR1B P49286 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4718899 0.91 CYP11B2 (0.44) CYP11B1CYP11B2GRM7HTR2AHTR2C
SCHEMBL4719266 0.90 LRRK2 (0.33) CYP11B1CYP11B2LRRK2GRM7ALPL
SCHEMBL14101738 0.90 LRRK2 (0.33) CYP11B1CYP11B2LRRK2GRM7ALPL
SCHEMBL4764976 0.90 CNR1 (0.34) CYP11B1CYP11B2LRRK2GRM7KDM4E
SCHEMBL4722103 0.89 L3MBTL1 (0.35) GRM7ALDH1A1ALPLALPIMAPT
SCHEMBL4724987 0.87 F10 (0.40) LRRK2ALDH1A1MAPTF10
SCHEMBL4724951 0.85 NTRK1 (0.32) LRRK2GRM7NTRK1MAPT
SCHEMBL4721216 0.85 F10 (0.32) LRRK2ALPLALPIMAPTF10
SCHEMBL4719764 0.85 PDE4A (0.41) CYP11B1CYP11B2GRM7WDR5KDM4E
SCHEMBL4722852 0.83 GRIN1 (0.34) NTRK1GRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed