SCHEMBL4764976

SCHEMBL4764976

COc1cc(OC)cc(-c2nn(-c3cc(Cl)ccc3C(F)(F)F)c(=O)c3c2CCN3)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 2/20 0.34
PTGS2 P35354 6/20 0.33
LRRK2 Q5S007 1/20 0.33
BRAF P15056 2/20 0.33
KDM4E B2RXH2 1/20 0.33
PTGS1 P23219 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
TSHR P16473 1/20 0.32
CYP2C19 P33261 1/20 0.32
THPO P40225 1/20 0.32
BLM P54132 1/20 0.32
PMP22 Q01453 1/20 0.32
HIF1A Q16665 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
GRM7 Q14831 1/20 0.32
CNR2 P34972 1/20 0.32
GABRP O00591 1/20 0.32
GABRD O14764 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4720876 0.90 CYP11B1 (0.33) LRRK2KDM4EGRM7NTRK1ALPL
SCHEMBL4719266 0.89 LRRK2 (0.33) LRRK2GRM7NTRK1ALPLALPI
SCHEMBL14101738 0.89 LRRK2 (0.33) LRRK2GRM7NTRK1ALPLALPI
SCHEMBL4722103 0.88 L3MBTL1 (0.35) CNR1GRM7CNR2ALPLALPI
SCHEMBL4724987 0.86 F10 (0.40) LRRK2
SCHEMBL4724951 0.84 NTRK1 (0.32) LRRK2GRM7NTRK1
SCHEMBL4721216 0.84 F10 (0.32) LRRK2ALPLALPI
SCHEMBL4718926 0.82 F10 (0.32) GRM7
SCHEMBL4724753 0.82 BRAF (0.33) BRAFKDM4ECYP1A2CYP3A4CYP2C9
SCHEMBL4718899 0.81 CYP11B2 (0.44) CYP1A2CYP3A4CYP2C9CYP2C19GRM7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed