SCHEMBL4723968

SCHEMBL4723968

Clc1cccc(CCCn2ccc3cncnc32)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 2/20 0.41
CTSL P07711 1/20 0.41
CTSS P25774 1/20 0.41
NOS3 P29474 1/20 0.41
NOS2 P35228 1/20 0.41
CYP1A2 P05177 4/20 0.40
CYP2C9 P11712 3/20 0.40
USP2 O75604 2/20 0.40
ALDH1A1 P00352 2/20 0.40
CYP2C19 P33261 2/20 0.40
CYP2D6 P10635 1/20 0.40
HSD17B10 Q99714 2/20 0.39
NTRK1 P04629 1/20 0.38
MAOA P21397 2/20 0.38
MAOB P27338 2/20 0.38
TAAR1 Q96RJ0 1/20 0.37
JAK2 O60674 2/20 0.37
HDAC6 Q9UBN7 2/20 0.37
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28212072 0.84 CYP1A2 (0.45) CYP1A2CYP2C9USP2ALDH1A1CYP2C19
SCHEMBL4763970 0.79 FGFR1 (0.40) CTSLCTSSMAOAMAOBTAAR1
SCHEMBL4723966 0.78 CYP1A2 (0.43) CYP1A2CYP2C9USP2ALDH1A1CYP2C19
SCHEMBL28212561 0.76 CYP1A2 (0.47) CYP1A2CYP2C9USP2ALDH1A1CYP2C19
SCHEMBL2173797 0.70 MKNK2 (0.40) CYP1A2CYP2C9USP2ALDH1A1CYP2C19
SCHEMBL25818492 0.70 MKNK2 (0.40) CYP1A2CYP2C9USP2ALDH1A1CYP2C19
SCHEMBL13195335 0.70 MKNK2 (0.40) CYP1A2
SCHEMBL15833488 0.68 MAPK13 (0.39) NOS1NOS3ALDH1A1HDAC6
SCHEMBL15833690 0.68 MTNR1A (0.36) ALDH1A1TAAR1
SCHEMBL28309924 0.67 KLKB1 (0.38) CYP1A2CYP2C9USP2ALDH1A1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957488-A1 3-AMINO-2-ARYLPROPYL AZAINDOLES AND USES THEREOF F.HOFFMANN-LA ROCHE AG (CH) 2008-08-20 EP disclosed
WO-2007062998-A1 3-AMINO-2-ARYLPROPYL AZAINDOLES AND USES THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2007-06-07 WO disclosed