SCHEMBL28212072

SCHEMBL28212072

c1ccc(CCCn2ccc3cncnc32)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 8/20 0.45
CYP2C19 P33261 8/20 0.45
CYP3A4 P08684 7/20 0.45
CYP2C9 P11712 7/20 0.45
ALDH1A1 P00352 6/20 0.45
TSHR P16473 4/20 0.45
CYP2D6 P10635 4/20 0.42
USP2 O75604 3/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
HSD17B10 Q99714 1/20 0.41
PLA2G7 Q13093 1/20 0.41
MAPK1 P28482 2/20 0.40
SIGMAR1 Q99720 1/20 0.39
LMNA P02545 3/20 0.39
KDM4E B2RXH2 1/20 0.39
POLB P06746 1/20 0.39
LTA4H P09960 1/20 0.38
CNOT7 Q9UIV1 1/20 0.38
ADORA2A P29274 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28212561 0.91 CYP1A2 (0.47) CYP1A2CYP2C19CYP3A4CYP2C9ALDH1A1
SCHEMBL4723968 0.84 NOS1 (0.41) CYP1A2CYP2C19CYP3A4CYP2C9ALDH1A1
SCHEMBL4723966 0.81 CYP1A2 (0.43) CYP1A2CYP2C19CYP3A4CYP2C9ALDH1A1
SCHEMBL25818492 0.75 MKNK2 (0.40) CYP1A2CYP2C19CYP3A4CYP2C9ALDH1A1
SCHEMBL2173797 0.75 MKNK2 (0.40) CYP1A2CYP2C19CYP3A4CYP2C9ALDH1A1
SCHEMBL13195335 0.75 MKNK2 (0.40) CYP1A2ADORA2A
SCHEMBL15833488 0.73 MAPK13 (0.39) ALDH1A1SIGMAR1KDM4E
SCHEMBL15833690 0.73 MTNR1A (0.36) ALDH1A1
SCHEMBL24110604 0.72 HTR2C (0.47)
SCHEMBL5068124 0.72 MKNK2 (0.42) CYP1A2CYP2C19CYP3A4CYP2C9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108137497-A Bicyclic derivatives, process for their preparation and pharmaceutical compositions containing them 法国施维雅药厂 2018-06-08 CN disclosed