SCHEMBL472476

SCHEMBL472476

O=C1NC(=O)C(Sc2ccccc2)C(=O)N1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 3/20 0.51
MEN1 O00255 1/20 0.51
KDM4A O75164 1/20 0.51
TDP2 O95551 1/20 0.51
KMT2A Q03164 1/20 0.51
APOBEC3G Q9HC16 1/20 0.51
CRBN Q96SW2 2/20 0.47
DDB1 Q16531 1/20 0.47
MAPT P10636 4/20 0.40
ALDH1A1 P00352 3/20 0.40
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
HPGD P15428 2/20 0.37
POLB P06746 1/20 0.37
MMP2 P08253 1/20 0.35
MMP9 P14780 1/20 0.35
GSK3B P49841 1/20 0.34
F2 P00734 2/20 0.34
PRSS1 P07477 2/20 0.34
USP2 O75604 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7031749 0.76 CRBN (0.45) KDM4CMEN1KDM4ATDP2KMT2A
SCHEMBL6794976 0.69 MAOA (0.45) KDM4CCRBNDDB1MAPTALDH1A1
SCHEMBL1639992 0.67 MAPT (0.48) MEN1KMT2ACRBNDDB1MAPT
SCHEMBL5798857 0.67 DDB1 (0.70) CRBNDDB1SMN1; SMN2
SCHEMBL10407251 0.67 CRBN (0.44) MEN1KMT2ACRBNDDB1MAPT
SCHEMBL8304222 0.67 CA2 (0.50) CRBNDDB1MAPTALDH1A1MAOB
SCHEMBL10817885 0.66 GAA (0.49) KDM4CMEN1KDM4ATDP2KMT2A
SCHEMBL1334635 0.65 MAPT (0.46) MEN1KMT2ACRBNDDB1MAPT
SCHEMBL17294198 0.65 MAPT (0.46) MEN1KMT2ACRBNDDB1MAPT
SCHEMBL22612145 0.64 DDB1 (1.00) CRBNDDB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 94 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250250418-A1 MIXTURE FOR INHIBITING THE EMISSION OF ALDEHYDES FROM POLYURETHANE FOAM FOR AN EXTENDED PERIOD OF TIME HUNTSMAN PETROCHEMICAL LLC 2025-08-07 US claimed
EP-4508111-A1 MIXTURE FOR INHIBITING THE EMISSION OF ALDEHYDES FROM POLYURETHANE FOAM FOR AN EXTENDED PERIOD OF TIME Huntsman Petrochemical LLC (US) 2025-02-19 EP claimed
WO-2023200641-A1 MIXTURE FOR INHIBITING THE EMISSION OF ALDEHYDES FROM POLYURETHANE FOAM FOR AN EXTENDED PERIOD OF TIME HUNTSMAN PETROCHEMICAL LLC (US) 2023-10-19 WO claimed
US-20120270962-A1 POLYMERIZABLE COMPOSITIONS CONTAINING SALTS OF BARBITURIC ACID DERIVATIVES 3M INNOVATIVE PROPERTIES COMPANY 2012-10-25 US claimed
US-8236871-B2 Polymerizable compositions containing salts of barbituric acid derivatives 3M INNOVATIVE PROPERTIES COMPANY (US) 2012-08-07 US claimed
EP-1881010-B1 Polymerizable compositions containing salts of barbituric acid derivatives 3M INNOVATIVE PROPERTIES CO (US) 2010-08-11 EP claimed
WO-2009100367-A2 COMPOSITIONS COMPRISING TOPICAL DPD INHIBITORS AND METHODS OF USING SAME IN THE TREATMENT OF HAND-FOOT SYNDROME ADHEREX TECHNOLOGIES INC. (CA) 2009-08-13 WO claimed
US-20090196833-A1 COMPOSITIONS COMPRISING TOPICAL DPD INHIBITORS AND METHODS OF USING SAME IN THE TREATMENT OF HAND-FOOT SYNDROME ADHEREX TECHNOLOGIES INC. (CA) 2009-08-06 US claimed
US-20090192239-A1 POLYMERIZABLE COMPOSITIONS CONTAINING SALTS OF BARBITURIC ACID DERIVATIVES SOLVENTUM INTELLECTUAL PROPERTIES COMPANY 2009-07-30 US claimed
US-20080255168-A1 METHODS FOR ADMINISTERING DPD INHIBITORS IN COMBINATION WITH 5-FU AND 5-FU PRODRUGS ADHEREX TECHNOLOGIES, INC. (CA) 2008-10-16 US claimed
WO-2006060697-A9 METHODS FOR ADMINISTERING DPD INHIBITORS IN COMBINATION WITH 5-FU AND 5-FU PRODRUGS ADHEREX TECHNOLOGIES INC (CA) 2006-09-21 WO claimed
US-20060148753-A1 Methods for administering DPD inhibitors in combination with 5-FU and 5-FU prodrugs ADHEREX TECHNOLOGIES, INC. (CA) 2006-07-06 US claimed
WO-2006060697-A1 METHODS FOR ADMINISTERING DPD INHIBITORS IN COMBINATION WITH 5-FU AND 5-FU PRODRUGS ADHEREX TECHNOLOGIES, INC. (CA) 2006-06-08 WO claimed
US-RE37623-E1 PHENYLTHIO AND PHENYLSELENO PYRIMIDINE ANALOGS el Kouni, Mahmoud H. 2002-04-02 US claimed
EP-0725641-B1 NOVEL INHIBITORS OF URIDINE PHOSPHORYLASE (UrdPase) AND DIHYDROURACIL DEHYDROGENASE (DHUDase) EL KOUNI MAHMOUD H (US) 2000-12-13 EP claimed
US-5721241-A PYRIMIDINE COMPOUND USEFUL TO DISRUPT VIRAL, CANCER, FUNGAL, PARASITE OR BACTERIAL REPLICATION AND DIHYDROURACIL DEHYDROGENASE OR URIDINE PHOSPHORYLASE INHIBITORS el Kouni, Mahmoud H. (US) 1998-02-24 US claimed
EP-0725641-A4 1996-09-04 EP claimed
EP-0725641-A1 NOVEL ENZYME INHIBITORS, THEIR SYNTHESIS, AND METHODS FOR USE El Kouni, Mahmoud H. (US) 1996-08-14 EP claimed
US-5476855-A Pyrimidine analogs and nucleosides el Kouni, Mahmoud H. (US) 1995-12-19 US claimed
WO-1995012400-A1 NOVEL ENZYME INHIBITORS, THEIR SYNTHESIS, AND METHODS FOR USE UAB RESEARCH FOUNDATION (US) 1995-05-11 WO claimed