SCHEMBL6794976

SCHEMBL6794976

O=C1NC(=O)C(c2ccc(Sc3ccccc3)cc2)C(=O)N1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.45
MAOB P27338 2/20 0.45
CRBN Q96SW2 3/20 0.39
DDB1 Q16531 2/20 0.39
ALDH1A1 P00352 2/20 0.38
HPGD P15428 1/20 0.38
MAPT P10636 3/20 0.37
MAPK1 P28482 2/20 0.37
KDM4E B2RXH2 1/20 0.37
PKM P14618 1/20 0.37
NTSR1 P30989 1/20 0.37
KDM4C Q9H3R0 1/20 0.37
TDP1 Q9NUW8 1/20 0.36
MCL1 Q07820 2/20 0.36
BCL2 P10415 1/20 0.36
SLC6A4 P31645 1/20 0.35
EZH2 Q15910 1/20 0.35
LMNA P02545 1/20 0.34
TP53 P04637 1/20 0.34
CYP1A2 P05177 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1639992 0.82 MAPT (0.48) MAOAMAOBCRBNDDB1ALDH1A1
SCHEMBL17294198 0.81 MAPT (0.46) MAOAMAOBCRBNDDB1ALDH1A1
SCHEMBL6380971 0.75 KDM1A (0.51) MAOAMAOBCA2
SCHEMBL6381012 0.71 KDM4E (0.48) ALDH1A1HPGDMAPK1KDM4ETDP1
SCHEMBL6380792 0.71 MEN1 (0.48) CRBNDDB1ALDH1A1HPGDMAPT
SCHEMBL472475 0.71 MAPT (0.50) CRBNDDB1ALDH1A1HPGDMAPT
SCHEMBL31579572 0.71 HAO1 (0.59) MAOBALDH1A1HPGDMAPTKDM4E
SCHEMBL4629140 0.70 PTPN1 (0.45) CRBNDDB1ALDH1A1HPGDMAPT
SCHEMBL31579581 0.70 TSHR (0.46) CRBNDDB1ALDH1A1TP53CA2
SCHEMBL11167420 0.70 MAPT (0.45) ALDH1A1MAPTMAPK1LMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6716845-B2 Barbituric acid derivatives HOFFMANN-LA ROCHE INC. 2004-04-06 US disclosed