SCHEMBL4724817

SCHEMBL4724817

CCNc1cc(-c2cc(C)cc(-c3cnco3)c2)nn(-c2cc(N3CCOCC3=O)ccc2C(F)(F)F)c1=O

nearest known ligand 0.33

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
F10 P00742 7/20 0.33
MAP4K1 Q92918 5/20 0.33
PIK3CD O00329 2/20 0.33
PIK3CA P42336 2/20 0.33
PIK3CG P48736 2/20 0.33
PIK3CB P42338 1/20 0.33
CMA1 P23946 2/20 0.32
LRRK2 Q5S007 1/20 0.31
RAF1 P04049 1/20 0.30
BRAF P15056 1/20 0.30
PTGS2 P35354 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
NTRK1 P04629 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4724965 0.91 FFAR1 (0.33)
SCHEMBL4721381 0.91 IMPDH2 (0.34) PIK3CDPIK3CAPIK3CGPIK3CBRAF1
SCHEMBL4724185 0.90 F10 (0.32) F10
SCHEMBL4719237 0.88 CMA1 (0.31) CMA1NTRK1
SCHEMBL4724962 0.88 JAK3 (0.33)
SCHEMBL4720665 0.86 PTK2 (0.31)
SCHEMBL4720659 0.86 PTK2 (0.31)
SCHEMBL4718681 0.86
SCHEMBL4723056 0.86 LMNA (0.32)
SCHEMBL4719688 0.85 GHSR (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed