SCHEMBL4724753

SCHEMBL4724753

COC(=O)CCNc1ccc(C(F)(F)F)c(-n2nc(-c3cc(OC)cc(OC)c3)c3c(c2=O)NCC3)c1

nearest known ligand 0.33

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BRAF P15056 4/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
SCD O00767 3/20 0.33
NTRK1 P04629 1/20 0.32
HTR2C P28335 3/20 0.32
HTR2B P41595 3/20 0.32
ATM Q13315 1/20 0.32
F10 P00742 1/20 0.31
HTR2A P28223 2/20 0.30
CYP1A2 P05177 2/20 0.30
KDM4E B2RXH2 1/20 0.30
KMT2A Q03164 1/20 0.30
ALDH1A1 P00352 1/20 0.30
CYP3A4 P08684 1/20 0.30
GAA P10253 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4724929 0.90 SCD (0.32) BRAFSCDNTRK1HTR2CHTR2B
SCHEMBL4723445 0.87 SMN1; SMN2 (0.35) BRAFSMN1; SMN2SCDHTR2CHTR2B
SCHEMBL4720876 0.83 CYP11B1 (0.33) NTRK1HTR2CHTR2BF10HTR2A
SCHEMBL4764976 0.82 CNR1 (0.34) BRAFNTRK1CYP1A2KDM4ECYP3A4
SCHEMBL14101738 0.82 LRRK2 (0.33) NTRK1F10
SCHEMBL4719266 0.82 LRRK2 (0.33) NTRK1F10
SCHEMBL4722572 0.81 PDE4A (0.37) SMN1; SMN2SCDCYP1A2KDM4EKMT2A
SCHEMBL4722103 0.81 L3MBTL1 (0.35) KMT2AALDH1A1GAA
SCHEMBL4722266 0.80 PDE4A (0.36) SMN1; SMN2SCDF10KDM4EKMT2A
SCHEMBL4721347 0.80 PDE4A (0.34) SMN1; SMN2SCDHTR2CHTR2BF10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed