SCHEMBL4763963

SCHEMBL4763963

CCN(CC)C(=O)C1CCc2[nH]c3ccccc3c2C1

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NR2E1 Q9Y466 1/20 0.52
SLC2A1 P11166 1/20 0.48
HSD17B10 Q99714 3/20 0.47
KDM4E B2RXH2 2/20 0.47
CYP1A2 P05177 2/20 0.47
CYP2D6 P10635 2/20 0.47
CYP2C9 P11712 2/20 0.47
CYP2C19 P33261 2/20 0.47
MAPK1 P28482 1/20 0.47
HPGD P15428 2/20 0.46
TP53 P04637 1/20 0.46
MAPT P10636 2/20 0.45
ALDH1A1 P00352 1/20 0.45
GAA P10253 1/20 0.45
ALOX15 P16050 1/20 0.45
HTR1B P28222 1/20 0.44
KMT2A Q03164 1/20 0.44
LMNA P02545 1/20 0.44
BAZ2B Q9UIF8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29059312 0.83 NR2E1 (0.50) NR2E1HSD17B10KDM4ECYP1A2CYP2D6
SCHEMBL31078247 0.81 KDM4E (0.64) NR2E1SLC2A1HSD17B10KDM4ECYP1A2
SCHEMBL4727252 0.81 KDM4E (0.64) NR2E1SLC2A1HSD17B10KDM4ECYP1A2
SCHEMBL31078488 0.81 NR2E1 (0.64) NR2E1HSD17B10KDM4ECYP1A2CYP2D6
SCHEMBL31078875 0.81 NR2E1 (0.60) NR2E1HSD17B10KDM4ECYP1A2CYP2D6
SCHEMBL12660565 0.81 NR2E1 (0.60) NR2E1HSD17B10KDM4ECYP1A2CYP2D6
SCHEMBL4903024 0.81 NR2E1 (0.64) NR2E1HSD17B10KDM4ECYP1A2CYP2D6
SCHEMBL2309545 0.81 NR2E1 (0.60) NR2E1HSD17B10KDM4ECYP1A2CYP2D6
SCHEMBL4725539 0.80 KMT2A (0.49) NR2E1SLC2A1HSD17B10KDM4ECYP1A2
SCHEMBL4728062 0.80 KDM4E (0.63) NR2E1HSD17B10KDM4ECYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1994022-A2 N-SUBSTITUTED-AZACYCLYLAMINES AS HISTAMINE-3 ANTAGONISTS Wyeth a Corporation of the State of Delaware (US) 2008-11-26 EP disclosed
WO-2007108936-A2 N-SUBSTITUTED-AZACYCLYLAMINES AS HISTAMINE-3 ANTAGONISTS WYETH (US) 2007-09-27 WO disclosed