SCHEMBL4727258

SCHEMBL4727258

CC(C)(C)NCC(O)COc1cccc2[nH]c3ccccc3c12

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 9/20 0.73
DNM1 Q05193 2/20 0.73
TLR4 O00206 4/20 0.67
DRD2 P14416 3/20 0.64
KMT2A Q03164 3/20 0.64
ADRB1 P08588 3/20 0.64
KDM4E B2RXH2 3/20 0.64
MAPT P10636 3/20 0.64
ADRB3 P13945 3/20 0.64
TDP1 Q9NUW8 2/20 0.64
SLC22A2 O15244 1/20 0.64
SLC22A1 O15245 1/20 0.64
MLNR O43193 1/20 0.64
NR1I2 O75469 1/20 0.64
KCNK2 O95069 1/20 0.64
ABCB11 O95342 1/20 0.64
APP P05067 1/20 0.64
ABCB1 P08183 1/20 0.64
HTR1A P08908 1/20 0.64
ADRA2A P08913 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13043810 0.90 ADRB2 (0.69) ADRB2DNM1TLR4DRD2KMT2A
SCHEMBL8295862 0.89 ADRB2 (0.67) ADRB2DNM1TLR4DRD2KMT2A
SCHEMBL7269307 0.88 ADRB2 (0.66) ADRB2DNM1TLR4DRD2KMT2A
SCHEMBL11339462 0.87 ADRB2 (0.65) ADRB2DNM1TLR4DRD2KMT2A
SCHEMBL3002063 0.86 ADRB2 (0.78) ADRB2DNM1TLR4DRD2KMT2A
SCHEMBL9258048 0.86 ADRB2 (0.64) ADRB2DNM1TLR4DRD2KMT2A
Carazolol SCHEMBL77901 0.84 ADRB2 (1.00) ADRB2DNM1TLR4DRD2KMT2A
Carazolol SCHEMBL6511163 0.84 ADRB2 (1.00) ADRB2DNM1TLR4DRD2KMT2A
Carazolol SCHEMBL29354289 0.84 ADRB2 (1.00) ADRB2DNM1TLR4DRD2KMT2A
Carazolol SCHEMBL77903 0.84 ADRB2 (1.00) ADRB2DNM1TLR4DRD2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021552-A9 BIASED LIGANDS AND METHODS OF IDENTIFYING SAME UNIV DUKE (US) 2008-05-29 WO claimed
WO-2008021552-A2 BIASED LIGANDS AND METHODS OF IDENTIFYING SAME DUKE UNIVERSITY (US) 2008-02-21 WO claimed