SCHEMBL4728237

SCHEMBL4728237

N[C@@H](Cc1ccc(F)cc1)CN1Cc2ccccc2C1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 5/20 0.51
SLC6A3 Q01959 4/20 0.51
HTR1A P08908 2/20 0.45
DRD2 P14416 2/20 0.45
HTR2A P28223 2/20 0.45
HTR7 P34969 2/20 0.45
HRH1 P35367 2/20 0.45
DRD3 P35462 2/20 0.45
HTR2B P41595 2/20 0.45
KDM4E B2RXH2 2/20 0.43
HSD17B10 Q99714 1/20 0.43
SLC6A2 P23975 2/20 0.42
DPP8 Q6V1X1 2/20 0.41
HDAC8 Q9BY41 4/20 0.40
EPHX1 P07099 1/20 0.40
MAPK1 P28482 2/20 0.40
HTT P42858 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
DPP7 Q9UHL4 2/20 0.39
DPP4 P27487 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4730009 0.87 EPHX1 (0.55) SLC6A4SLC6A3SLC6A2HDAC8EPHX1
SCHEMBL30239684 0.84 DPP4 (0.44) SLC6A4SLC6A3DRD2DPP8DPP7
SCHEMBL3191528 0.73 SLC6A4 (0.58) SLC6A4EPHX1DPP7DPP4
SCHEMBL17732253 0.73 SIGMAR1 (0.42) KDM4EMAPK1HTT
SCHEMBL4779114 0.73 SLC6A4 (0.55) SLC6A4SLC6A3HTR1ADRD2DRD3
SCHEMBL495855 0.72 HDAC8 (0.50) HDAC8EPHX1CARM1
SCHEMBL29724812 0.71 KDM4E (0.47) SLC6A4SLC6A3HTR1ADRD2HTR2A
Hydrochloric Acid SCHEMBL496040 0.71 HDAC8 (0.51) HDAC8EPHX1CARM1
SCHEMBL1529725 0.71 CASP3 (0.57) SLC6A4SLC6A3HSD17B10TSHR
SCHEMBL1529723 0.71 CASP3 (0.57) SLC6A4SLC6A3HSD17B10TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008036308-A2 AMINO-SUBSTITUTED HETEROCYCLES, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH SIGNAL PHARMACEUTICALS, LLC (US) 2008-03-27 WO disclosed