SCHEMBL4728295

SCHEMBL4728295

COc1ccc(-c2cc(N)cnc2C)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.50
MAPT P10636 3/20 0.49
DYRK1A Q13627 2/20 0.46
PTGS2 P35354 2/20 0.46
MAPK1 P28482 2/20 0.46
TP53 P04637 1/20 0.46
TSHR P16473 1/20 0.46
HTT P42858 1/20 0.46
MAPK10 P53779 1/20 0.46
PTK2B Q14289 1/20 0.46
NCOA1 Q15788 1/20 0.46
NCOA3 Q9Y6Q9 1/20 0.46
MAP4K4 O95819 1/20 0.45
CHEK2 O96017 1/20 0.45
NPC1 O15118 3/20 0.44
RAB9A P51151 3/20 0.44
TDP1 Q9NUW8 1/20 0.44
FYN P06241 1/20 0.43
ABL1 P00519 1/20 0.43
DRD1 P21728 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28722185 0.85 CHEK2 (0.59) KMT2AMAPTDYRK1APTGS2MAPK1
SCHEMBL14293715 0.81 DRD1 (0.56) KMT2AMAPTMAPK1TP53TSHR
SCHEMBL17178235 0.80 ALDH1A1 (0.55) KMT2AMAPTMAPK1TP53HTT
SCHEMBL14923566 0.79 IRAK4 (0.46) KMT2AMAPTMAPK1TP53TSHR
SCHEMBL24171393 0.78 FYN (0.47) MAP4K4CHEK2FYNABL1KIT
SCHEMBL11236122 0.77 FYN (0.45) FYNABL1DRD1
SCHEMBL4728311 0.77 ABL1 (0.50) KMT2AMAPTMAPK1TP53NPC1
SCHEMBL4727538 0.74 KAT2B (0.49) KMT2AMAPTMAPK1HTTNPC1
SCHEMBL5904303 0.73 CHEK2 (0.58) KMT2AMAPTDYRK1AMAPK1TP53
SCHEMBL415914 0.73 TDP1 (0.58) KMT2AMAPTDYRK1AMAPK1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021388-A1 HETEROARYL DERIVATIVES AS CYTOKINE INHIBITORS KEMIA, INC. (US) 2008-02-21 WO disclosed