SCHEMBL4729157

SCHEMBL4729157

NC(=O)CNC(c1ccc2ccccc2n1)c1ccc2ccccc2n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
KDM4C Q9H3R0 1/20 0.42
HDAC8 Q9BY41 2/20 0.41
HSD17B10 Q99714 1/20 0.40
KDM4E B2RXH2 2/20 0.40
S1PR3 Q99500 2/20 0.40
MGAM O43451 1/20 0.40
CYP1A2 P05177 1/20 0.40
LMNA P02545 1/20 0.40
PKM P14618 1/20 0.40
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9870690 0.75 MGAM (0.48) ALDH1A1GAAMAPTHDAC8HSD17B10
SCHEMBL7375731 0.74 ALDH1A1 (0.44) ALDH1A1GAAMAPTKDM4CHDAC8
SCHEMBL10605297 0.73 HDAC6 (0.52) ALDH1A1GAAMAPTKDM4CHSD17B10
SCHEMBL29457163 0.71 CYP1A2 (0.47) ALDH1A1GAAMAPTHDAC8HSD17B10
SCHEMBL4725705 0.71 HDAC1 (0.51) ALDH1A1GAAMAPTKDM4CHDAC8
SCHEMBL7527822 0.70 GRM7 (0.54) ALDH1A1GAACYP1A2LMNAPKM
SCHEMBL27721065 0.69 MGAM (0.50) ALDH1A1GAAMAPTKDM4CHDAC8
SCHEMBL5721000 0.69 KDM4E (0.46) ALDH1A1GAAMAPTKDM4CHDAC8
SCHEMBL5720996 0.69 KDM4E (0.46) ALDH1A1GAAMAPTKDM4CHDAC8
SCHEMBL29858224 0.69 KDM4E (0.53) ALDH1A1GAAMAPTHSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021745-A2 HEPATITIS C VIRUS ENTRY INHIBITORS ITHERX PHARMACEUTICALS, INC. (US) 2008-02-21 WO disclosed
US-6399631-B1 3-AMIDO OR 3-SULFONAMIDO; EATING DISORDERS IN HUMANS, DOGS AND CATS PFIZER INC. 2002-06-04 US disclosed