SCHEMBL7375731

SCHEMBL7375731

[CH2]C(CC(N)=O)c1ccc2ccccc2n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
HSD17B10 Q99714 1/20 0.44
GAA P10253 1/20 0.44
MAPT P10636 1/20 0.44
MGAM O43451 1/20 0.41
CYP1A2 P05177 1/20 0.41
KDM4E B2RXH2 3/20 0.41
LMNA P02545 1/20 0.41
PKM P14618 1/20 0.41
PRNP P04156 3/20 0.39
RXFP1 Q9HBX9 3/20 0.39
MEN1 O00255 1/20 0.38
HPGD P15428 1/20 0.38
KMT2A Q03164 1/20 0.38
CNR2 P34972 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
NCF1 P14598 1/20 0.38
NOS2 P35228 1/20 0.38
BACE1 P56817 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9870690 0.76 MGAM (0.48) ALDH1A1HSD17B10GAAMAPTMGAM
SCHEMBL4729157 0.74 ALDH1A1 (0.46) ALDH1A1HSD17B10GAAMAPTMGAM
SCHEMBL5721000 0.73 KDM4E (0.46) ALDH1A1HSD17B10GAAMAPTMGAM
SCHEMBL5720996 0.73 KDM4E (0.46) ALDH1A1HSD17B10GAAMAPTMGAM
SCHEMBL29457163 0.72 CYP1A2 (0.47) ALDH1A1HSD17B10GAAMAPTMGAM
SCHEMBL4064465 0.72 ALDH1A1 (0.50) ALDH1A1HSD17B10GAAMAPTMGAM
SCHEMBL7462368 0.70 IDO1 (0.53) ALDH1A1CYP1A2LMNAKMT2A
SCHEMBL10069400 0.69 ALDH1A1 (0.48) ALDH1A1HSD17B10GAAMAPTMGAM
SCHEMBL29057277 0.69 CYP1A2 (0.42) ALDH1A1HSD17B10GAAMAPTMGAM
SCHEMBL20746476 0.69 NCF1 (0.43) ALDH1A1HSD17B10MAPTMGAMCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165500-A1 AMIDE DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEINASES,TNF-ALPHA,AND AGGRECANASE Du Pont Pharmaceuticals Company (US) 2002-01-02 EP disclosed
WO-2000059874-A1 NOVEL AMIDE DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEINASES, TNF-α, AND AGGRECANASE DU PONT PHARMACEUTICALS COMPANY (US) 2000-10-12 WO disclosed