SCHEMBL4729660

SCHEMBL4729660

CCC(C)(C)C(=O)Nc1cc(N2CCOCC2)c2ccccc2n1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MOK Q9UQ07 1/20 0.53
NCF1 P14598 2/20 0.53
CNR2 P34972 6/20 0.53
PDE10A Q9Y233 1/20 0.49
USP2 O75604 1/20 0.48
CNR1 P21554 2/20 0.48
ALDH1A1 P00352 2/20 0.47
MAPT P10636 2/20 0.47
METAP1 P53582 1/20 0.46
PIK3R1 P27986 1/20 0.45
PIK3CA P42336 1/20 0.45
MTOR P42345 1/20 0.45
KDM4E B2RXH2 1/20 0.45
HIF1A Q16665 1/20 0.45
PKM P14618 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
HSD17B10 Q99714 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4730661 0.99 MOK (0.52) MOKNCF1CNR2PDE10AUSP2
SCHEMBL4732598 0.84 CNR2 (0.65) MOKCNR2CNR1
SCHEMBL4731636 0.84 ALDH1A1 (0.56) MOKNCF1PDE10AUSP2ALDH1A1
SCHEMBL4733439 0.77 NPSR1 (0.59) MOKNCF1USP2ALDH1A1MAPT
SCHEMBL4732942 0.75 MOK (0.51) MOKNCF1CNR2PDE10AUSP2
SCHEMBL5241851 0.72 NCF1 (0.64) MOKNCF1USP2ALDH1A1MAPT
SCHEMBL5093588 0.70 NCF1 (1.00) NCF1USP2ALDH1A1MAPTMETAP1
SCHEMBL4731630 0.70 NCF1 (0.55) MOKNCF1USP2ALDH1A1MAPT
SCHEMBL19475310 0.70 MOK (0.77) MOKNCF1ALDH1A1MAPTMETAP1
SCHEMBL19475531 0.69 MOK (1.00) MOKPDE10AALDH1A1MAPTPIK3R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008063625-A2 PYRIDINE COMPOUNDS AND METHODS OF THEIR USE ADOLOR CORPORATION (US) 2008-05-29 WO claimed
WO-2008063625-A2 PYRIDINE COMPOUNDS AND METHODS OF THEIR USE ADOLOR CORPORATION (US) 2008-05-29 WO disclosed
WO-2008063625-A2 PYRIDINE COMPOUNDS AND METHODS OF THEIR USE ADOLOR CORPORATION (US) 2008-05-29 WO disclosed