SCHEMBL4730146

SCHEMBL4730146

O=C(O)NCC(=O)NC1CCN(Cc2ccccc2)CC1

nearest known ligand 0.75

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 16/20 0.75
KMT2A Q03164 1/20 0.71
DRD4 P21917 1/20 0.66
POLB P06746 1/20 0.65
L3MBTL1 Q9Y468 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7268908 0.89 SIGMAR1 (0.79) SIGMAR1POLBL3MBTL1
SCHEMBL4840680 0.88 CCR2 (0.76) SIGMAR1KMT2ADRD4
Hydrochloric Acid SCHEMBL29640479 0.88 SIGMAR1 (0.77) SIGMAR1POLBL3MBTL1
SCHEMBL5862113 0.86 SIGMAR1 (1.00) SIGMAR1
SCHEMBL2425554 0.86 SIGMAR1 (0.78) SIGMAR1KMT2ADRD4POLBL3MBTL1
SCHEMBL3075354 0.85 SIGMAR1 (0.81) SIGMAR1POLBL3MBTL1
SCHEMBL5124505 0.85 SIGMAR1 (0.81) SIGMAR1POLBL3MBTL1
SCHEMBL29640480 0.85 SIGMAR1 (0.81) SIGMAR1POLBL3MBTL1
Hydrochloric Acid SCHEMBL21410212 0.84 SIGMAR1 (0.76) SIGMAR1KMT2ADRD4POLBL3MBTL1
SCHEMBL6177317 0.83 SIGMAR1 (0.79) SIGMAR1POLBL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008032036-A1 6-BENZIMIDAZ0LYL-2-M0RPH0LIN0-4- (AZETIDINE, PYRROLIDINE, PIPERIDINE OR AZEPINE) PYRIMIDINE DERIVATIVES AS PI3K AND MTOR INHIBITORS FOR THE TREATMENT OF PROLIFERATIVE DISORDERS ASTRAZENECA AB (SE) 2008-03-20 WO disclosed