SCHEMBL4731059

SCHEMBL4731059

COC(=O)C(CSCc1csc(-c2cccc(-c3cccc4c3oc3ccccc34)c2)n1)NC(=O)OC(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 3/20 0.36
PPARA Q07869 3/20 0.36
CCR2 P41597 1/20 0.36
GSTP1 P09211 1/20 0.36
GSTM2 P28161 1/20 0.36
PTPRB P23467 1/20 0.36
NFKB1 P19838 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
PPARD Q03181 2/20 0.35
GGPS1 O95749 1/20 0.35
SHMT1 P34896 1/20 0.35
ALDH1A1 P00352 3/20 0.34
MAPT P10636 3/20 0.34
KLK5 Q9Y337 1/20 0.34
KDM4E B2RXH2 1/20 0.34
GAA P10253 1/20 0.34
PKM P14618 1/20 0.34
HPGD P15428 1/20 0.34
ALOX12 P18054 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4730467 0.93 PPARG (0.44) PPARGPPARACCR2PTPRBPPARD
SCHEMBL14260809 0.93 PPARG (0.44) PPARGPPARACCR2PTPRBPPARD
SCHEMBL14260756 0.89 CCR2 (0.36) PPARGPPARACCR2PTPRBGGPS1
SCHEMBL4728145 0.88 PPARG (0.47) PPARGPPARAPTPRBPPARDGAA
SCHEMBL14260755 0.88 PPARG (0.47) PPARGPPARAPTPRBPPARDGAA
SCHEMBL3866879 0.81 PPARA (0.50) PPARGPPARAGSTP1GSTM2NFKB1
SCHEMBL3866499 0.81 PPARA (0.50) PPARGPPARAGSTP1GSTM2NFKB1
SCHEMBL13897379 0.81 GSTP1 (0.42) PPARGPPARAGSTP1GSTM2NFKB1
SCHEMBL3871194 0.81 GSTP1 (0.42) PPARGPPARAGSTP1GSTM2NFKB1
SCHEMBL4730121 0.78 P2RY12 (0.37) PPARGPPARAMAPTGAAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008033934-A1 SUBSTITUTED HETEROARYL CARBOXYLIC ACID DERIVATIVES AS PTB-1B INHIBITORS THE INSTITUTES FOR PHARMACEUTICAL DISCOVERY, LLC (US) 2008-03-20 WO disclosed