SCHEMBL4731075

SCHEMBL4731075

Nc1ccc(-c2nc(N3CCOCC3)cc(C3(C(F)F)Nc4ccccc4N3)n2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.49
MTOR P42345 4/20 0.48
PIK3CA P42336 3/20 0.48
PIK3R1 P27986 1/20 0.48
ATR Q13535 2/20 0.47
NPSR1 Q6W5P4 3/20 0.46
MAPT P10636 2/20 0.46
TSHR P16473 1/20 0.46
MAPK1 P28482 1/20 0.46
HSD17B10 Q99714 1/20 0.46
KMT2A Q03164 2/20 0.45
MEN1 O00255 1/20 0.45
CYP1A2 P05177 3/20 0.41
CYP3A4 P08684 3/20 0.41
CYP2C9 P11712 3/20 0.41
CYP2C19 P33261 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
LMNA P02545 1/20 0.41
PIK3CD O00329 1/20 0.40
ALDH1A1 P00352 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4730536 0.89 ATR (0.43) HTTMTORPIK3CAATRNPSR1
SCHEMBL4727905 0.87 ATR (0.49) HTTMTORPIK3CAATRNPSR1
SCHEMBL4727055 0.83 PIK3CA (0.41) HTTMTORPIK3CAATRNPSR1
SCHEMBL4794320 0.82 PIK3CA (0.48) HTTMTORPIK3CAPIK3R1NPSR1
SCHEMBL4730594 0.79 AKT1 (0.44) MTORPIK3CAPIK3R1ATRPIK3CD
SCHEMBL4731787 0.78 JAK2 (0.45) MTORPIK3CAATRMAPTKMT2A
SCHEMBL4727870 0.77 PIK3CB (0.48) MTORPIK3CAATRNPSR1TSHR
SCHEMBL4726457 0.77 PIK3CB (0.48) MTORPIK3CAATRNPSR1TSHR
SCHEMBL4728682 0.74 TERT (0.43) MTORPIK3CAATRCYP3A4PIK3CD
SCHEMBL3719793 0.73 MAPT (0.84) HTTMTORPIK3CAPIK3R1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008032077-A1 PYRIMIDINE DERIVATIVES ASTRAZENECA AB (SE) 2008-03-20 WO disclosed