SCHEMBL4731378

SCHEMBL4731378

CC(C)(C)[SiH2]OC(C)(C)c1cccc(-c2cnc(N)c(C=O)n2)c1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.41
PIK3CA P42336 1/20 0.41
PIK3CG P48736 1/20 0.41
ATR Q13535 11/20 0.36
PRKDC P78527 2/20 0.33
TYRO3 Q06418 2/20 0.33
LDHB P07195 2/20 0.32
MAP4K4 O95819 1/20 0.32
LDHA P00338 1/20 0.32
ASIC3 Q9UHC3 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
NEK2 P51955 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4731377 0.73 ATR (0.40) PIK3CDPIK3CAPIK3CGATRPRKDC
SCHEMBL19672862 0.68 HSP90AA1 (0.51) ATR
SCHEMBL23732958 0.65 ATR (0.32) ATRPRKDC
SCHEMBL14312975 0.64 PIK3CD (0.44) PIK3CDPIK3CAPIK3CG
SCHEMBL3463003 0.62 LDHA (0.58) ATRLDHBMAP4K4LDHA
SCHEMBL4783565 0.62 PRKCI (0.43)
SCHEMBL1166675 0.62 ADORA2A (0.41)
SCHEMBL840466 0.61 ESR1 (0.39)
SCHEMBL3124960 0.61 ACHE (0.35)
SCHEMBL1167036 0.61 GSK3B (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008038010-A1 PYRAZINE DERIVATIVES AND THEIR USE IN THERAPY VERNALIS (R & D) LIMITED (GB) 2008-04-03 WO disclosed