SCHEMBL4731382

SCHEMBL4731382

COCC(C)Nc1cc(-c2ccc(-c3cc4ncccn4n3)cc2)sc1C(=O)OC

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.41
MAPT P10636 5/20 0.41
ALDH1A1 P00352 2/20 0.41
LMNA P02545 1/20 0.41
HPGD P15428 2/20 0.40
HTT P42858 1/20 0.39
ATM Q13315 1/20 0.39
NPSR1 Q6W5P4 2/20 0.38
TP53 P04637 2/20 0.38
KMT2A Q03164 1/20 0.38
RXFP1 Q9HBX9 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4143220 0.90 MAPT (0.45) KDM4EMAPTALDH1A1LMNAHPGD
SCHEMBL1728318 0.82 MAPT (0.55) KDM4EMAPTALDH1A1LMNAHPGD
SCHEMBL4779360 0.81 MAPT (0.62) KDM4EMAPTALDH1A1LMNAHPGD
SCHEMBL1458894 0.80 KDM4E (0.41) KDM4EMAPTALDH1A1LMNAHPGD
SCHEMBL14291019 0.78 KDM4E (0.36) KDM4EHPGDHTTATM
SCHEMBL4755031 0.77 KDM4E (0.61) KDM4EMAPTALDH1A1LMNAHPGD
SCHEMBL4755035 0.77 KDM4E (0.61) KDM4EMAPTALDH1A1LMNAHPGD
SCHEMBL4793397 0.77 KDM4E (0.36) KDM4EMAPTALDH1A1LMNAHPGD
SCHEMBL4793400 0.77 KDM4E (0.36) KDM4EMAPTALDH1A1LMNAHPGD
SCHEMBL3262134 0.76 PLA2G2A (0.36) KDM4EMAPTALDH1A1LMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008043791-A2 THIOPHENE DERIVATIVES FOR TREATING HEPATITIS C SMITHKLINE BEECHAM CORPORATION (US) 2008-04-17 WO disclosed
WO-2008043791-A2 THIOPHENE DERIVATIVES FOR TREATING HEPATITIS C SMITHKLINE BEECHAM CORPORATION (US) 2008-04-17 WO disclosed