SCHEMBL4793397

SCHEMBL4793397

COCC(COC)N(c1cc(-c2ccc(-c3cc4ncccn4n3)cc2)sc1C(=O)OC)C(=O)[C@H]1CC[C@H](C)CC1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.36
HTT P42858 1/20 0.36
ATM Q13315 1/20 0.36
PDE4D Q08499 5/20 0.35
SYK P43405 4/20 0.34
SLC6A9 P48067 1/20 0.31
HPGD P15428 1/20 0.31
IKBKB O14920 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4793400 1.00 KDM4E (0.36) KDM4EHTTATMPDE4DSYK
SCHEMBL4777606 0.94 IKBKB (0.34) KDM4EHTTATMPDE4DSYK
SCHEMBL4725145 0.94 IKBKB (0.34) KDM4EHTTATMPDE4DSYK
SCHEMBL14291019 0.94 KDM4E (0.36) KDM4EHTTATMPDE4DSYK
SCHEMBL4140069 0.91 KDM4E (0.38) KDM4EHTTATMPDE4DSYK
SCHEMBL4140062 0.91 KDM4E (0.38) KDM4EHTTATMPDE4DSYK
SCHEMBL14291286 0.88 IKBKB (0.33) PDE4DSYKSLC6A9IKBKB
SCHEMBL4795076 0.88 ALDH1A1 (0.38) KDM4EHTTATMPDE4DSYK
SCHEMBL4795067 0.88 ALDH1A1 (0.38) KDM4EHTTATMPDE4DSYK
SCHEMBL4155397 0.87 KDM4E (0.38) KDM4EHTTATMPDE4DSYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008017688-A1 2-CARBOXY THIOPHENE DERIVATIVES AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2008-02-14 WO disclosed
WO-2008017688-A1 2-CARBOXY THIOPHENE DERIVATIVES AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2008-02-14 WO disclosed