SCHEMBL4732047

SCHEMBL4732047

Nc1c(Br)cc(CCO)cc1Br

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.46
MAPT P10636 2/20 0.46
CA2 P00918 3/20 0.38
CA1 P00915 2/20 0.38
CA9 Q16790 2/20 0.38
CA3 P07451 1/20 0.38
GSK3B P49841 1/20 0.38
CA12 O43570 1/20 0.38
CA4 P22748 1/20 0.38
CA6 P23280 1/20 0.38
CA5A P35218 1/20 0.38
CA7 P43166 1/20 0.38
CA14 Q9ULX7 1/20 0.38
CA5B Q9Y2D0 1/20 0.38
TDP1 Q9NUW8 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
ALOX5 P09917 1/20 0.37
BACE1 P56817 1/20 0.37
ADRB2 P07550 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11505357 0.85 MAPT (0.55) GAAMAPTCA2CA1CA9
SCHEMBL21633076 0.81 ADRB2 (0.46) GAAMAPTCA2CA1CA9
SCHEMBL2925262 0.78 TDP1 (0.48) GAAMAPTCA2CA1CA9
SCHEMBL32669352 0.77 CA2 (0.32) GAAMAPTCA2CA1CA9
SCHEMBL4734190 0.76 TDP1 (0.37) GAAMAPTCA2CA1CA9
SCHEMBL7871857 0.76 MAPT (0.46) GAAMAPTCA2CA1CA9
SCHEMBL10980722 0.76 GAA (0.46) GAAMAPTCA2CA1CA9
SCHEMBL3085307 0.76 KDM4E (0.47) GAAMAPTCA2CA1CA9
SCHEMBL11372198 0.74 THRA (0.53) CA2CA1GSK3BTHRATHRB
SCHEMBL5981517 0.74 MAPT (0.55) GAAMAPTCA2CA1CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008053158-A1 INHIBITORS OF P38 MITOGEN-ACTIVATED PROTEIN KINASE CHROMA THERAPEUTICS LTD. (GB) 2008-05-08 WO disclosed
WO-2008053158-A1 INHIBITORS OF P38 MITOGEN-ACTIVATED PROTEIN KINASE CHROMA THERAPEUTICS LTD. (GB) 2008-05-08 WO disclosed
US-6099625-A Ink composition ZENECA LIMITED (GB) 2000-08-08 US disclosed