SCHEMBL4732058

SCHEMBL4732058

CCOc1ccc(C(=O)N2CCC(NS(=O)(=O)c3ccc(C(C)C)cc3C(F)(F)F)CC2)cn1

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SFRP1 Q8N474 18/20 0.51
KDM4E B2RXH2 1/20 0.40
HSD17B10 Q99714 1/20 0.40
WNT3 P56703 5/20 0.40
MGLL Q99685 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4734093 0.89 SFRP1 (0.53) SFRP1KDM4EHSD17B10WNT3
SCHEMBL4734362 0.87 SFRP1 (0.64) SFRP1WNT3MGLL
SCHEMBL4733149 0.79 SFRP1 (0.48) SFRP1WNT3
SCHEMBL4738622 0.76 SFRP1 (0.61) SFRP1WNT3
SCHEMBL4733299 0.76 SFRP1 (0.64) SFRP1
SCHEMBL4731611 0.75 SFRP1 (0.69) SFRP1WNT3
SCHEMBL4735241 0.75 SFRP1 (0.62) SFRP1WNT3
SCHEMBL4737077 0.75 SFRP1 (0.68) SFRP1WNT3
SCHEMBL4786060 0.75 SFRP1 (0.69) SFRP1WNT3
SCHEMBL4735995 0.74 SFRP1 (0.63) SFRP1WNT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008061016-A1 N-SUBSTITUTED PIPERIDINYL 4 -ARYLSULFONAMIDES AS MODULATORS OF THE SECRETED FRIZZLED RELATED PROTEIN- 1 WYETH (US) 2008-05-22 WO claimed
WO-2008061016-A1 N-SUBSTITUTED PIPERIDINYL 4 -ARYLSULFONAMIDES AS MODULATORS OF THE SECRETED FRIZZLED RELATED PROTEIN- 1 WYETH (US) 2008-05-22 WO disclosed