SCHEMBL4733115

SCHEMBL4733115

Fc1ccc2c(c1)Sc1ccc(OC(F)(F)F)cc1C2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR3 P46089 4/20 0.42
PPM1A P35813 1/20 0.34
TRPV4 Q9HBA0 2/20 0.33
CES1 P23141 1/20 0.33
TRPA1 O75762 1/20 0.32
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
GMNN O75496 1/20 0.32
USP2 O75604 1/20 0.32
LMNA P02545 1/20 0.32
TP53 P04637 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
GAA P10253 1/20 0.32
CYP2C9 P11712 1/20 0.32
PKM P14618 1/20 0.32
ALOX15 P16050 1/20 0.32
NFKB1 P19838 1/20 0.32
SLC6A2 P23975 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4733314 0.74 RAD52 (0.44) NPC1RAB9ALMNATP53CYP1A2
SCHEMBL11182451 0.74 ALDH1A1 (0.41) GAASLC6A2SLC6A3SLC6A4KIF11
SCHEMBL29756225 0.74 NOX1 (0.38) LMNABLMPIM1
Ammonia Solution, Strong SCHEMBL2438706 0.72 GPR3 (0.46) GPR3CES1NPC1RAB9AGMNN
SCHEMBL4733543 0.69 GPR3 (0.40) GPR3PPM1ATRPV4CES1TRPA1
SCHEMBL4733537 0.69 GPR3 (0.40) GPR3PPM1ATRPV4CES1TRPA1
SCHEMBL20014448 0.69 GPR3 (0.36) GPR3CES1NPC1RAB9AGMNN
SCHEMBL5905690 0.69 KMT2A (0.59) GPR3CES1LMNAGAABLM
SCHEMBL11346578 0.66 MAPK14 (0.43) NPC1RAB9ALMNA
SCHEMBL5535809 0.66 NOX1 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008061029-A1 ARYL SULFONAMIDE DERIVATIVES AND METHODS OF THEIR USE WYETH (US) 2008-05-22 WO disclosed