SCHEMBL4733537

SCHEMBL4733537

O=S1(=O)c2ccc(OC(F)(F)F)cc2Cc2ccc(F)cc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR3 P46089 3/20 0.40
CES1 P23141 1/20 0.34
GALR1 P47211 2/20 0.34
SLC40A1 Q9NP59 1/20 0.34
CTSL P07711 1/20 0.34
TRPV4 Q9HBA0 2/20 0.34
MAOA P21397 1/20 0.33
BACE1 P56817 1/20 0.33
ABL1 P00519 1/20 0.32
PSEN1 P49768 1/20 0.32
PSEN2 P49810 1/20 0.32
APH1B Q8WW43 1/20 0.32
NCSTN Q92542 1/20 0.32
APH1A Q96BI3 1/20 0.32
PSENEN Q9NZ42 1/20 0.32
HSD11B1 P28845 1/20 0.32
KIF11 P52732 1/20 0.31
TRPA1 O75762 1/20 0.31
PPM1A P35813 1/20 0.31
TRPV1 Q8NER1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4733543 0.84 GPR3 (0.40) GPR3CES1CTSLTRPV4BACE1
SCHEMBL4732228 0.76 MAOA (0.37) MAOAPSEN1PSEN2APH1BNCSTN
SCHEMBL4730918 0.74 GPR3 (0.39) GPR3CES1GALR1SLC40A1CTSL
SCHEMBL4730132 0.73 CYP17A1 (0.39) MAOA
Ammonia Solution, Strong SCHEMBL2438706 0.70 GPR3 (0.46) GPR3CES1BACE1KIF11TRPV1
SCHEMBL4733115 0.69 GPR3 (0.42) GPR3CES1CTSLTRPV4BACE1
SCHEMBL11823803 0.68 AKR1C3 (0.40) MAOAPSEN1PSEN2APH1BNCSTN
SCHEMBL4733982 0.64 HTR2A (0.35) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL13932523 0.63 MAOA (0.44) MAOA
SCHEMBL4730920 0.63 GPR3 (0.39) GPR3TRPV4PPM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008061029-A1 ARYL SULFONAMIDE DERIVATIVES AND METHODS OF THEIR USE WYETH (US) 2008-05-22 WO disclosed