SCHEMBL4733307

SCHEMBL4733307

CC(=O)C(CBr)c1ccc(F)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.44
ESR2 Q92731 1/20 0.44
PTPN1 P18031 1/20 0.42
HTT P42858 1/20 0.40
HDAC3 O15379 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC10 Q969S8 1/20 0.40
HDAC11 Q96DB2 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
HDAC9 Q9UKV0 1/20 0.40
HDAC5 Q9UQL6 1/20 0.40
ALDH1A1 P00352 2/20 0.37
KDM4E B2RXH2 1/20 0.37
FFAR1 O14842 1/20 0.37
AOC3 Q16853 1/20 0.37
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27483504 0.84 PTPN1 (0.45) PTPN1HTTHDAC3HDAC4HDAC1
SCHEMBL16055955 0.82 ESR1 (0.46) ESR1ESR2ALDH1A1LMNA
SCHEMBL12073123 0.82 PTPN1 (0.44) PTPN1HDAC3HDAC4HDAC1HDAC7
SCHEMBL16149256 0.81 GABBR2 (0.46) ESR1ESR2HTTHDAC3HDAC4
SCHEMBL2002439 0.80 CYP2C19 (0.44) ESR1ESR2ALDH1A1LMNA
SCHEMBL2739002 0.78 ESR1 (0.42) ESR1ESR2HTTHDAC3HDAC4
SCHEMBL9756750 0.77 ESR1 (0.41) ESR1ESR2HTTHDAC3HDAC4
SCHEMBL12167815 0.75 ESR1 (0.40) ESR1ESR2HTTHDAC3HDAC4
SCHEMBL684103 0.75 ADRB2 (0.49) ESR1ESR2HTTHDAC3HDAC4
SCHEMBL684740 0.75 AOC3 (0.40) ESR1ESR2HTTHDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008054454-A2 NITROGEN-CONTAINING HETEROCYCLE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS, AND METHODS OF USE THEREOF AS ANTIVIRAL AGENTS TRANSTECH PHARMA, INC. (US) 2008-05-08 WO disclosed